Josef Jampilek
Selected publications of:
  1. Jampilek J, Dolezal M, Opletalova V, Hartl J. 5-Lipoxygenase, Leukotrienes Biosynthesis and Potential Antileukotrienic Agents. Curr Med Chem. 2006;13(2):117–129.
  2. Musiol R, Jampilek J, Buchta V, Silva L, Niedbala H, Podeszwa B, Palka A, et al. Antifungal Properties of New Series of Quinoline Derivatives. Bioorg Med Chem. 2006;14(10):3592–3598.
  3. Vinsova, J, Cermakova K, Tomeckova A, Ceckova M, Jampilek J, Cermak P, Kunes J, et al. Synthesis and Antimicrobial Evaluation of New 2-Substituted 5,7-Di-tertbutylbenzoxazoles. Bioorg Med Chem. 2006;14(17):5850–5865.
  4. Musiol R, Jampilek J, Kralova K, Richardson DR, Kalinowski D, Podeszwa B, Finster J, et al. Investigating Biological Activity Spectrum for Novel Quinoline Analogues. Bioorg Med Chem. 2007;15(3):1280–1288.
  5. Imramovsky A, Polanc S, Vinsova J, Kocevar, M, Jampilek J, Reckova Z, Kaustova J. A New Modification of Antitubercular Active Molecules. Bioorg Med Chem. 2007;15(7):2551–2559.
  6. Jampilek J, Brychtova K. Azone Analogues: Classification, Design, and Transdermal Penetration Principles. Med Res Rev. 2012;32 (5):907–947.
  7. Culen M, Rezacova A, Jampilek J, Dohnal J. Designing a Dynamic Dissolution Method: A Review of Instrumental Options and Corresponding Physiology of Stomach and Small Intestine. J Pharm Sci. 2013;102(9):2995–3017.
  8. Jampilek J. Recent Advances in Design of Potential Quinoxaline Anti-Infectives. Curr Med Chem. 2014;21(38):4347–4373.
  9. Zadrazilova I, Pospisilova S, Masarikova M, Imramovsky A, Monreal-Ferriz J, Vinsova J, Cizek A, et al. Salicylanilide Carbamates: Promising Antibacterial Agents with High In Vitro Activity against Methicillin-resistant Staphylococcus aureus (MRSA). Eur J Pharm Sci. 2015;77:197–207.
  10. Kos J, Zadrazilova I, Nevin E, Soral M, Gonec T, Kollar P, Oravec M. Coffey A, O'Mahony J, Liptaj T, Kralova K, Jampilek J. Ring-substituted 8-Hydroxyquinoline-2-carboxanilides as Potential Antimycobacterial Agents. Bioorg Med Chem. 2015;23, in press, DOI:10.1016/j.bmc.2015.06.047.